SCHEMBL28110985

SCHEMBL28110985

Nc1nc(Cc2ccccc2)nc2[nH]ccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
ADORA1 P30542 2/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
CDC7 O00311 1/20 0.41
DBF4 Q9UBU7 1/20 0.41
CSF1R P07333 1/20 0.40
DHPS P49366 1/20 0.39
HTR6 P50406 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
APP P05067 1/20 0.39
LTB4R Q15722 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30297934 0.86 HTR6 (0.40) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL29715845 0.86 APP (0.41) CYP2D6ADORA1ADORA2AADORA2BCDC7
Hydrochloric Acid SCHEMBL30297929 0.85 HTR6 (0.39) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL30298043 0.84 HRH4 (0.46) CYP1A2CYP3A4CYP2D6CYP2C9ADORA1
SCHEMBL20508793 0.84 HRH4 (0.46) CYP1A2CYP3A4CYP2D6CYP2C9ADORA1
Hydrochloric Acid SCHEMBL30297964 0.83 HRH4 (0.44) CYP1A2CYP2D6ADORA1ADORA2AHRH4
SCHEMBL30910330 0.81 L3MBTL1 (0.44) CYP1A2CYP3A4CYP2C9CYP2C19CDC7
SCHEMBL29246448 0.81 L3MBTL1 (0.44) CYP1A2CYP3A4CYP2C9CYP2C19CDC7
SCHEMBL20508772 0.80 ADORA1 (0.45) ADORA1ADORA2AADORA2BHTR6DYRK1A
SCHEMBL20508822 0.80 PDE8B (0.39) ADORA1ADORA2AHRH4DYRK1ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061973-A Pyrrolo [2,3-D ] pyrimidinyl, pyrrolo [2,3-B ] pyrazinyl and pyrrolo [2,3-D ] pyridylacrylamide 辉瑞公司 2016-10-26 CN disclosed