SCHEMBL28111092

SCHEMBL28111092

CCC(C)C(NC(=O)OC(C)(C)C)C(=O)Oc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.53
CTSK P43235 1/20 0.53
ALDH1A1 P00352 3/20 0.49
MAPT P10636 2/20 0.49
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CA2 P00918 2/20 0.47
KDM4E B2RXH2 2/20 0.46
KMT2A Q03164 1/20 0.46
SYK P43405 1/20 0.46
HPGD P15428 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PSENEN Q9NZ42 1/20 0.45
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
HTT P42858 1/20 0.45
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12890771 0.87 KLK5 (0.51) CTSSCTSKALDH1A1MAPTKDM4E
SCHEMBL30471370 0.87 KLK5 (0.51) CTSSCTSKALDH1A1MAPTKDM4E
SCHEMBL24390653 0.84 CYP3A4 (0.59) CTSSCTSKMAPTRAB9ACA2
SCHEMBL12214475 0.84 CYP3A4 (0.59) CTSSCTSKMAPTRAB9ACA2
SCHEMBL26226843 0.83 ALDH1A1 (0.67) CTSSCTSKALDH1A1MAPTRAB9A
SCHEMBL22137002 0.83 ALDH1A1 (0.67) CTSSCTSKALDH1A1MAPTRAB9A
SCHEMBL16284648 0.83 ALDH1A1 (0.67) CTSSCTSKALDH1A1MAPTRAB9A
SCHEMBL27817322 0.83 KDM4E (0.53) CTSSCTSKALDH1A1MAPTKDM4E
SCHEMBL28232199 0.81 CYP1A2 (0.54) CTSSALDH1A1MAPTRAB9ACTSL
SCHEMBL11802988 0.81 CTSS (0.49) CTSSCTSKALDH1A1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307772-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2024-06-28 CN disclosed
CN-113307772-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-08-27 CN disclosed
CN-106257976-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-02-02 CN disclosed
CN-106257976-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2016-12-28 CN disclosed