SCHEMBL28111509

SCHEMBL28111509

COC(=O)C(C)(CC=O)C(C)=O

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.34
MAPT P10636 1/20 0.33
ALDH1A1 P00352 1/20 0.31
GAA P10253 2/20 0.30
MGAM O43451 1/20 0.30
SI P14410 1/20 0.30
MGAM2 Q2M2H8 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3174371 0.89 DGAT1 (0.38) DGAT1MAPTPKM
SCHEMBL27886351 0.83 DGAT1 (0.34) DGAT1MAPTPKM
SCHEMBL365038 0.76 DGAT1 (0.38) DGAT1MAPTPKM
SCHEMBL556529 0.76 DGAT1 (0.38) DGAT1ALDH1A1GAAMGAMSI
SCHEMBL6229413 0.74 TSHR (0.37) DGAT1MAPTALDH1A1GAAMGAM
SCHEMBL8899156 0.74 TSHR (0.37) DGAT1MAPTALDH1A1GAAMGAM
SCHEMBL12138536 0.73 DGAT1 (0.34) DGAT1ALDH1A1PKM
SCHEMBL30343873 0.73 DGAT1 (0.34) DGAT1MAPTALDH1A1
SCHEMBL3183165 0.72 DGAT1 (0.35) DGAT1PKM
SCHEMBL1422494 0.72 DGAT1 (0.35) DGAT1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106132967-B Compound as ROS1 inhibitor 詹森药业有限公司 2019-05-28 CN disclosed
CN-106132967-A 4,5,6,7 tetrahydro-pyrazoles being replaced also [1,5 a] pyrimidine derivatives and 2,3 dihydro 1H imidazo [1,2 b] pyrazole derivatives as ROS1 inhibitor 詹森药业有限公司 2016-11-16 CN disclosed