SCHEMBL28111983

SCHEMBL28111983

CCCCc1cncc(C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 7/20 0.51
HCAR2 Q8TDS4 4/20 0.50
POLB P06746 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
ALDH1A1 P00352 5/20 0.49
KDM4E B2RXH2 4/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
LMNA P02545 2/20 0.49
MAPT P10636 2/20 0.49
NFKB1 P19838 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
PKM P14618 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
THPO P40225 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2516239 0.95 RARB (0.53) RARBHCAR2POLBCYP2C9CYP2C19
SCHEMBL2566879 0.93 RARB (0.55) RARBHCAR2POLBCYP2C9CYP2C19
SCHEMBL846393 0.82 CYP2C9 (0.61) HCAR2POLBCYP2C9CYP2C19ALDH1A1
SCHEMBL30281282 0.82 CYP2C9 (0.61) HCAR2POLBCYP2C9CYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL20719501 0.81 KDM4E (0.49) HCAR2POLBCYP2C9CYP2C19ALDH1A1
SCHEMBL2530451 0.80 GPR84 (0.44) RARBALDH1A1MEN1KMT2ANFKB1
SCHEMBL2513768 0.80 GPR84 (0.44) RARBALDH1A1MEN1KMT2AMAPT
SCHEMBL9701286 0.80 RARB (0.59) RARBALDH1A1KDM4EMEN1KMT2A
SCHEMBL914005 0.80 RARB (0.59) RARBALDH1A1KDM4EMEN1KMT2A
Butane SCHEMBL11036256 0.79 CYP2C9 (0.67) HCAR2POLBCYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106470993-A The azepine quinazoline inhibitor of Atypical protein kinase C 癌症研究科技有限公司 2017-03-01 CN disclosed