SCHEMBL28112274

SCHEMBL28112274

CCC(=O)c1ncc(C2CC2)s1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 10/20 0.37
CDK2 P24941 10/20 0.37
CDK5 Q00535 10/20 0.37
CDK5R1 Q15078 1/20 0.37
SMYD3 Q9H7B4 2/20 0.33
PLAT P00750 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.31
RAB9A P51151 2/20 0.31
NPC1 O15118 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16266936 0.79 ALDH1A1 (0.39) CCNE1CDK2CDK5CDK5R1SMN1; SMN2
SCHEMBL8833248 0.73 CCNE1 (0.36) CCNE1CDK2CDK5CDK5R1SMN1; SMN2
SCHEMBL25801701 0.73 SMYD3 (0.40) SMYD3SMN1; SMN2RAB9ANPC1GAA
SCHEMBL31595821 0.72 GSK3B (0.37) GAA
SCHEMBL24572410 0.69 CCNE1 (0.49) CCNE1CDK2CDK5CDK5R1SMN1; SMN2
SCHEMBL8833517 0.68 CDK2 (0.33) CCNE1CDK2CDK5CDK5R1
SCHEMBL24572407 0.68 CCNE1 (0.45) CCNE1CDK2CDK5CDK5R1SMN1; SMN2
SCHEMBL8833766 0.67 CCNE1 (0.35) CCNE1CDK2CDK5CDK5R1SMN1; SMN2
SCHEMBL11937013 0.67 MAPT (0.37)
SCHEMBL8833251 0.66 SMN1; SMN2 (0.35) CCNE1CDK2CDK5CDK5R1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106068265-A Dihydropyridone MGAT2 inhibitors for the treatment of metabolic disorders 百时美施贵宝公司 2016-11-02 CN disclosed