SCHEMBL28114427

SCHEMBL28114427

FC(F)(F)COC[C@@H]1CCCN1Cc1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
POLB P06746 2/20 0.48
HRH3 Q9Y5N1 1/20 0.44
CHRNB2 P17787 3/20 0.44
CHRNA4 P43681 3/20 0.44
CHRNA7 P36544 2/20 0.42
CHRNA1 P02708 1/20 0.42
CHRNB1 P11230 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNB3 Q05901 1/20 0.42
CHRM2 P08172 2/20 0.40
CHRM1 P11229 2/20 0.40
CHRM3 P20309 2/20 0.40
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
MDM2 Q00987 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28114428 1.00 KDM4E (0.48) KDM4EPOLBHRH3CHRNB2CHRNA4
SCHEMBL14779735 0.85 FAAH (0.50)
SCHEMBL14779737 0.85 FAAH (0.50)
SCHEMBL27958431 0.82 KDM4E (0.56) KDM4EPOLBHRH3CHRNB2CHRNA4
SCHEMBL27958432 0.82 KDM4E (0.56) KDM4EPOLBHRH3CHRNB2CHRNA4
SCHEMBL14780344 0.81 CHRNB2 (0.42) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL14780346 0.81 CHRNB2 (0.42) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL21937561 0.77 KDM4E (0.60) KDM4EPOLBHRH3CHRNB2CHRNA4
SCHEMBL4310630 0.75 FAAH (0.53) KDM4EPOLBCHRNB2CHRNA4CHRNA7
SCHEMBL4310635 0.75 FAAH (0.53) KDM4EPOLBCHRNB2CHRNA4CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103814021-B Dihydroquinoline 2 ketone derivatives 霍夫曼-拉罗奇有限公司 2016-12-21 CN disclosed