SCHEMBL28114733

SCHEMBL28114733

COc1cc(C(=O)c2ccc(Br)c(OC)c2)ccc1Br

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.72
CYP1A2 P05177 2/20 0.68
CYP2C19 P33261 2/20 0.68
TSHR P16473 2/20 0.68
CYP3A4 P08684 1/20 0.68
CYP2C9 P11712 1/20 0.68
SLC22A6 Q4U2R8 1/20 0.63
SLC22A8 Q8TCC7 1/20 0.63
CYP2D6 P10635 1/20 0.62
HPGD P15428 1/20 0.62
GAA P10253 1/20 0.58
HTT P42858 3/20 0.56
LMNA P02545 2/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
TUBB4A P04350 4/20 0.53
TUBB P07437 4/20 0.53
TUBA3C P0DPH7 4/20 0.53
TUBA1B P68363 4/20 0.53
TUBA4A P68366 4/20 0.53
TUBB4B P68371 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31164292 0.91 CYP1A2 (0.77) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL1129401 0.91 CYP1A2 (0.77) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL12982799 0.86 LMNA (0.55) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL644265 0.86 CA12 (0.69) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL29688674 0.86 LMNA (0.55) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL17786825 0.85 ALDH1A1 (0.53) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL426745 0.85 MAPT (0.62) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL432016 0.85 TSHR (0.62) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL27630437 0.84 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4
SCHEMBL27026756 0.83 MAPT (0.53) ALDH1A1CYP1A2CYP2C19TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104114552-B Substituted Triazolopyridine and the purposes as TTK inhibitor thereof 拜耳知识产权有限责任公司 2016-12-28 CN disclosed