SCHEMBL28114877

SCHEMBL28114877

COc1cccc(CNc2ccnc(Cl)n2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 14/20 0.61
CYP1A2 P05177 6/20 0.61
CYP3A4 P08684 6/20 0.61
CYP2D6 P10635 6/20 0.61
CYP2C19 P33261 6/20 0.61
LMNA P02545 6/20 0.61
TSHR P16473 5/20 0.61
MEN1 O00255 3/20 0.61
KMT2A Q03164 3/20 0.61
ALDH1A1 P00352 3/20 0.61
MAPK1 P28482 3/20 0.61
ALOX15 P16050 2/20 0.61
TP53 P04637 1/20 0.61
DYRK1A Q13627 5/20 0.61
MAPT P10636 4/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
USP2 O75604 2/20 0.61
CYP2C9 P11712 2/20 0.61
TDP1 Q9NUW8 1/20 0.61
HSD17B10 Q99714 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13504222 0.83 CLK4 (0.68) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4554748 0.82 MAP4K4 (0.54) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL15917642 0.80 CLK4 (0.45) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL20511459 0.79 MAPT (0.57) CLK4TSHRMEN1KMT2AALDH1A1
SCHEMBL30268041 0.78 CYP1A2 (0.56) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL1666752 0.78 CYP1A2 (0.64) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL2518146 0.78 CCNK (0.56) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL3452299 0.78 CYP1A2 (0.69) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4861102 0.78 CYP1A2 (0.56) CLK4CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL5752435 0.78 CYP1A2 (0.56) CLK4CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104262263-B N,6 diphenylpyrimidine-4-amine Bcr-Abl inhibitors as well as preparation method and application thereof 西安交通大学 2017-01-11 CN disclosed