SCHEMBL28114887

SCHEMBL28114887

O=C(c1ccc(F)c(F)c1)N1CCNCC1.[PbH2]

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.65
MEN1 O00255 1/20 0.65
HSD11B1 P28845 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
HPGD P15428 1/20 0.51
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TDO2 P48775 1/20 0.48
DPP4 P27487 1/20 0.48
HRH4 Q9H3N8 2/20 0.48
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
ABL1 P00519 1/20 0.46
BCR P11274 1/20 0.46
PGR P06401 1/20 0.45
PARP1 P09874 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27986249 0.98 KMT2A (0.67) KMT2AMEN1HSD11B1SIGMAR1HPGD
SCHEMBL24746207 0.84 KMT2A (0.54) KMT2AMEN1HSD11B1SIGMAR1HPGD
SCHEMBL1018987 0.84 SIGMAR1 (0.53) KMT2AMEN1HSD11B1SIGMAR1HPGD
Hydrochloric Acid SCHEMBL623790 0.83 HPGD (0.55) KMT2AMEN1HSD11B1SIGMAR1HPGD
SCHEMBL421902 0.83 KMT2A (0.73) KMT2AMEN1HSD11B1HPGDALDH1A1
SCHEMBL2655426 0.83 KMT2A (0.73) KMT2AMEN1HSD11B1HPGDALDH1A1
SCHEMBL29944147 0.81 MEN1 (0.71) KMT2AMEN1HSD11B1HPGDALDH1A1
SCHEMBL226167 0.81 SIGMAR1 (0.56) KMT2AMEN1SIGMAR1HPGDTDO2
SCHEMBL8358137 0.80 SIGMAR1 (0.81) SIGMAR1HPGDALDH1A1MKNK1MKNK2
SCHEMBL2004712 0.80 KMT2A (0.69) KMT2AMEN1HSD11B1HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104262263-B N,6 diphenylpyrimidine-4-amine Bcr-Abl inhibitors as well as preparation method and application thereof 西安交通大学 2017-01-11 CN disclosed