SCHEMBL28114893

SCHEMBL28114893

Cc1ccccc1CC(CO)CO

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.43
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
DPP4 P27487 1/20 0.39
DPP7 Q9UHL4 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KCNH2 Q12809 1/20 0.38
HPGD P15428 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CTBP2 P56545 1/20 0.38
TSHR P16473 1/20 0.38
ACHE P22303 1/20 0.38
CHRM2 P08172 1/20 0.37
PTGS1 P23219 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29647878 0.90 TRPA1 (0.44) TAAR1PPARGPPARADPP4DPP7
SCHEMBL345975 0.90 TRPA1 (0.44) TAAR1PPARGPPARADPP4DPP7
SCHEMBL9817577 0.81 TRPA1 (0.42) TAAR1PPARGPPARASLC6A2SLC6A4
SCHEMBL27531705 0.81 CYP1A2 (0.50) TAAR1PPARGPPARASLC6A2SLC6A4
SCHEMBL8418317 0.81 CYP1A2 (0.50) TAAR1PPARGPPARASLC6A2SLC6A4
SCHEMBL20694193 0.80 TAAR1 (0.45) TAAR1PPARGPPARASLC6A2SLC6A4
SCHEMBL3935731 0.79 DPP4 (0.47) TAAR1PPARGPPARADPP4DPP7
SCHEMBL7997555 0.79 DPP4 (0.47) TAAR1PPARGPPARADPP4DPP7
SCHEMBL17101198 0.78 TAAR1 (0.54) TAAR1PPARGPPARADPP4DPP7
SCHEMBL13812287 0.77 TAAR1 (0.46) TAAR1PPARGPPARASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106103423-B Pyrazine compounds 阿斯利康(瑞典)有限公司 2019-12-06 CN disclosed
CN-106103423-A Chemical compound 阿斯利康(瑞典)有限公司 2016-11-09 CN disclosed