SCHEMBL28115058

SCHEMBL28115058

COC(=O)c1cnc2c(Br)cn(Br)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMD14 O00487 1/20 0.43
POLB P06746 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK10 P53779 2/20 0.40
PPARG P37231 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 3/20 0.40
ATM Q13315 1/20 0.40
KDM4E B2RXH2 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 2/20 0.38
HSD17B10 Q99714 1/20 0.36
USP2 O75604 1/20 0.36
NOTUM Q6P988 1/20 0.35
JMJD6 Q6NYC1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25385523 0.86 PSMD14 (0.43) PSMD14POLBALDH1A1MAPK10PPARG
SCHEMBL30314598 0.78 ALDH1A1 (0.40) PSMD14POLBALDH1A1MAPK10PPARG
SCHEMBL24050550 0.78 ALDH1A1 (0.40) PSMD14POLBALDH1A1MAPK10PPARG
SCHEMBL20951908 0.74 PSMD14 (0.43) PSMD14POLBALDH1A1MAPK10PPARG
SCHEMBL1505593 0.72 MAPK1 (0.53) PSMD14POLBALDH1A1MAPK10PPARG
SCHEMBL28115459 0.71 PSMD14 (0.43) PSMD14POLBALDH1A1KMT2AMAPK1
SCHEMBL20605105 0.71 PSMD14 (0.70) PSMD14POLBALDH1A1GAATSHR
SCHEMBL197929 0.70 MAPK1 (0.51) PSMD14POLBALDH1A1MAPK10PPARG
SCHEMBL30414233 0.70 MAPK1 (0.51) PSMD14POLBALDH1A1MAPK10PPARG
SCHEMBL335911 0.70 MAPK1 (0.51) PSMD14POLBALDH1A1MAPK10PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106117205-A Pyrazolo spiral shell ketone derivatives as S-acetyl-coenzyme-A carboxylase inhibitor class 辉瑞大药厂 2016-11-16 CN disclosed