SCHEMBL28115423

SCHEMBL28115423

O=CC1CCc2ccc(F)cc2N1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
PARP10 Q53GL7 1/20 0.36
HTR2C P28335 3/20 0.35
HTR2B P41595 2/20 0.35
HTR5A P47898 2/20 0.35
HTR2A P28223 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
KMT2A Q03164 2/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
SRD5A1 P18405 4/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28114067 0.89 ESR1 (0.36) PARP1PARP10HTR2CHTR2BHTR5A
SCHEMBL27771607 0.80 CA9 (0.47) KMT2AMAPTMEN1
SCHEMBL27825250 0.80 CMA1 (0.41) PARP1PARP10HTR2CHTR2BHTR2A
SCHEMBL27545193 0.80 ESR2 (0.43) ACHE
SCHEMBL1550271 0.77 MTNR1A (0.42) HTR2AMAPTNPC1
SCHEMBL30929595 0.77 MTNR1A (0.42) HTR2AMAPTNPC1
SCHEMBL27844296 0.76 GRIN2B (0.36) HTR2CHTR2BHTR2A
SCHEMBL22660299 0.75 FABP6 (0.39) TRPV1MAPT
SCHEMBL27844279 0.75 NPC1 (0.42) KMT2AMAPTMEN1NPC1
SCHEMBL13496703 0.75 HTR5A (0.36) PARP1PARP10HTR5AKMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103827101-B Dicyclo dihydroquinoline-2-ketone derivatives 霍夫曼-拉罗奇有限公司 2016-12-07 CN disclosed