SCHEMBL28115513

SCHEMBL28115513

Cc1cc(C(F)(F)F)c(CNC(=O)OC(C)(C)C)cn1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 1/20 0.51
CACNA1B Q00975 1/20 0.51
CACNA1C Q13936 1/20 0.51
EPHX2 P34913 4/20 0.41
AAK1 Q2M2I8 2/20 0.41
LMNA P02545 2/20 0.40
POLB P06746 1/20 0.40
KDM4A O75164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TRPV1 Q8NER1 2/20 0.38
RAF1 P04049 1/20 0.38
BRAF P15056 1/20 0.38
NTRK1 P04629 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NAMPT P43490 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3301163 0.85 KDM4A (0.41) CACNA1HCACNA1BCACNA1CAAK1LMNA
SCHEMBL16822059 0.83 EPHX2 (0.41) EPHX2POLBNTRK1MAPK1
SCHEMBL31380341 0.78 CACNA1H (0.47) CACNA1HCACNA1BCACNA1CAAK1LMNA
SCHEMBL20320534 0.77 LMNA (0.45) CACNA1HCACNA1BCACNA1CAAK1LMNA
SCHEMBL12656366 0.76 EPHX2 (0.46) CACNA1HCACNA1BCACNA1CEPHX2AAK1
SCHEMBL16094537 0.76 EPHX2 (0.46) CACNA1HCACNA1BCACNA1CEPHX2LMNA
SCHEMBL20380317 0.75 LMNA (0.59) CACNA1HCACNA1BCACNA1CEPHX2LMNA
SCHEMBL26101477 0.75 CACNA1H (0.45) CACNA1HCACNA1BCACNA1CEPHX2AAK1
SCHEMBL24821267 0.74 EPHX2 (0.44) CACNA1HCACNA1BCACNA1CEPHX2LMNA
SCHEMBL31431106 0.74 CACNA1H (0.47) CACNA1HCACNA1BCACNA1CAAK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106170290-A Substituted di-amino-pyrimidine based compound, combinations thereof and treatment method thereof 西格诺药品有限公司 2016-11-30 CN disclosed