SCHEMBL2811570

SCHEMBL2811570

CC(C)(O)C#Cc1cccc(O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.44
CA12 O43570 2/20 0.44
CA2 P00918 2/20 0.44
CA9 Q16790 2/20 0.44
CA1 P00915 1/20 0.44
HAO1 Q9UJM8 1/20 0.42
ASIC3 Q9UHC3 1/20 0.41
LMNA P02545 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 2/20 0.41
CA5A P35218 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CA14 Q9ULX7 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
FFAR1 O14842 2/20 0.41
MAP3K14 Q99558 1/20 0.40
EGFR P00533 1/20 0.40
ACHE P22303 2/20 0.39
HSD17B13 Q7Z5P4 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11443850 0.88 HAO1 (0.46) HAO1ASIC3LMNAMAP3K14EGFR
SCHEMBL2815252 0.86 GRM5 (0.45) GRM5CA12CA2CA9CA1
SCHEMBL2629434 0.81 GRM5 (0.49) GRM5HAO1ASIC3FFAR1MAP3K14
SCHEMBL19720165 0.79 GABRA1 (0.36) HAO1ASIC3LMNAALDH1A1CYP3A4
SCHEMBL24506081 0.79 HAO1 (0.41) HAO1ASIC3LMNAMAP3K14EGFR
SCHEMBL13692775 0.79 FFAR1 (0.42) CA12CA2CA9CA1HAO1
SCHEMBL30092382 0.79 MAP3K14 (0.45) CA12CA2CA9CA1HAO1
SCHEMBL1477501 0.79 KCNH2 (0.50) GRM5HAO1ASIC3MAP3K14EGFR
SCHEMBL1795798 0.79 PDK1 (0.43) GRM5HAO1ASIC3FFAR1MAP3K14
SCHEMBL471131 0.79 MAP3K14 (0.45) CA12CA2CA9CA1HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed
US-7291692-B2 Polyarylene oxide and method of producing the same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-11-06 US disclosed
US-20050096452-A1 Polyarylene oxide and method of producing the same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2005-05-05 US disclosed
US-4590304-A Protected ethynylated phenols THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1986-05-20 US disclosed
US-4540833-A Protected ethynylated phenols THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1985-09-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B GRM5 2797/4885CA12 2006/4885CA2 1282/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 GRM5 3664/4885CA12 610/4885CA2 831/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.