SCHEMBL28115935

SCHEMBL28115935

NC(=O)c1cnc(C(F)F)cn1.O=C(O)c1cnc(C(F)F)cn1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 2/20 0.47
ADORA3 P0DMS8 1/20 0.40
TSHR P16473 1/20 0.40
MC4R P32245 1/20 0.40
ADRA1A P35348 1/20 0.40
MC3R P41968 1/20 0.40
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 3/20 0.37
NAPRT Q6XQN6 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
ASPH Q12797 2/20 0.37
KDM8 Q8N371 1/20 0.37
P4HTM Q9NXG6 2/20 0.36
P4HA1 P13674 1/20 0.36
MIF P14174 1/20 0.36
BACE1 P56817 10/20 0.35
ALDH1A1 P00352 1/20 0.35
BACE2 Q9Y5Z0 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29447022 0.94 SIRT6 (0.52) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL15352404 0.94 SIRT6 (0.52) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL29447044 0.93 KDM4E (0.42) SIRT6KDM4ENAPRTHCAR2ASPH
SCHEMBL990507 0.93 KDM4E (0.42) SIRT6KDM4ENAPRTHCAR2ASPH
Trifluoroacetic Acid SCHEMBL30088405 0.88 SIRT6 (0.43) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL17712841 0.82 SIRT6 (0.64) SIRT6ADORA3TSHRMC4RADRA1A
2-Picolinic Acid SCHEMBL28871212 0.79 P4HTM (0.61) KMT2AKDM4ENAPRTHCAR2P4HTM
SCHEMBL15360279 0.78 KDM4E (0.39) SIRT6TSHRKMT2AKDM4ENAPRT
SCHEMBL2635320 0.76 SIRT6 (0.73) SIRT6ADORA3TSHRMC4RADRA1A
SCHEMBL2628913 0.76 SIRT6 (0.52) SIRT6ADORA3TSHRMC4RADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104245680-B Process for producing 5- (difluoromethyl) pyrazine-2-carboxylic acid and production intermediate thereof 卫材R&D管理有限公司 2016-11-23 CN disclosed