SCHEMBL28116633

SCHEMBL28116633

COc1cc(N2CCNC2)ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 5/20 0.53
TGFBR1 P36897 2/20 0.50
ACVR1 Q04771 2/20 0.50
HTR3E A5X5Y0 3/20 0.49
HTR3B O95264 3/20 0.49
HTR3A P46098 3/20 0.49
HTR3D Q70Z44 3/20 0.49
HTR3C Q8WXA8 3/20 0.49
ALK Q9UM73 1/20 0.48
BRD4 O60885 2/20 0.46
CHRNB2 P17787 2/20 0.46
CHRNA4 P43681 2/20 0.46
HTR1A P08908 2/20 0.46
HTR7 P34969 2/20 0.46
SIGMAR1 Q99720 2/20 0.45
SUV39H2 Q9H5I1 2/20 0.45
HTR1D P28221 1/20 0.44
HTR1B P28222 1/20 0.44
DRD2 P14416 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1639487 0.91 ADRB1 (0.65) ADRB1TGFBR1ACVR1HTR3EHTR3B
Hydrochloric Acid SCHEMBL1638699 0.89 ADRB1 (0.63) ADRB1TGFBR1ACVR1HTR3EHTR3B
Hydrochloric Acid SCHEMBL27692066 0.89 ADRB1 (0.63) ADRB1TGFBR1ACVR1HTR3EHTR3B
SCHEMBL1639658 0.78 BCL2A1 (0.50) ADRB1TGFBR1ACVR1ALKSUV39H2
SCHEMBL1639654 0.78 BCL2A1 (0.50) ADRB1TGFBR1ACVR1ALKSUV39H2
SCHEMBL2867159 0.78 BCL2A1 (0.50) ADRB1TGFBR1ACVR1ALKSUV39H2
SCHEMBL13456456 0.78 ALK (0.43) ADRB1TGFBR1ACVR1HTR3EHTR3B
SCHEMBL8182707 0.78 ADRB1 (0.65) ADRB1TGFBR1ACVR1HTR3EHTR3B
SCHEMBL13682933 0.78 ALDH1A1 (0.58) SUV39H2LMNAMAPT
SCHEMBL12625177 0.78 ALDH1A1 (0.58) SUV39H2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008375-B Tetrahydroimidazo [1,5-d ] [1,4] oxazepine derivatives 卫材R&D管理有限公司 2016-12-28 CN disclosed