SCHEMBL28117217

SCHEMBL28117217

CCOC(=O)CCCc1c[nH]c2ccc(Br)cc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
CYP2C19 P33261 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.70
SLC6A4 P31645 2/20 0.56
MTNR1A P48039 1/20 0.56
MTNR1B P49286 1/20 0.56
GABRA1 P14867 1/20 0.55
GABRB1 P18505 1/20 0.55
GABRA3 P34903 1/20 0.55
GABRB2 P47870 1/20 0.55
HTR2A P28223 1/20 0.52
TRPM8 Q7Z2W7 1/20 0.52
HTR1A P08908 2/20 0.52
ALDH1A1 P00352 2/20 0.51
GPR84 Q9NQS5 1/20 0.50
MPO P05164 3/20 0.49
PKM P14618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6220357 0.86 CYP2D6 (0.71) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL16433186 0.85 CYP1A2 (0.70) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7230859 0.85 CYP1A2 (0.70) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3703101 0.85 PKM (0.67) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8292283 0.84 CYP2D6 (0.68) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6222377 0.83 CYP2D6 (0.66) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9374131 0.82 SMN1; SMN2 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL27642166 0.82 SLC6A4 (0.60) CYP2C9CYP2C19SLC6A4MTNR1AMTNR1B
SCHEMBL31173807 0.82 SLC6A4 (0.60) CYP2C9CYP2C19SLC6A4MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL9369222 0.81 SMN1; SMN2 (0.97) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104163813-B Substituted indole compound, and preparation method and use thereof 广东东阳光药业有限公司 2017-02-01 CN disclosed