SCHEMBL28117984

SCHEMBL28117984

CC[CH]c1c(F)cc(C(F)(F)F)cc1F

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.42
IDO1 P14902 4/20 0.35
GAA P10253 1/20 0.33
TRPA1 O75762 3/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
CES2 O00748 1/20 0.32
CYP1A2 P05177 1/20 0.32
PTPN5 P54829 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
APP P05067 1/20 0.31
PTGS1 P23219 1/20 0.31
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18242800 0.80 CACNA1H (0.35) IDO1CES2PTPN5CYP3A4TSHR
SCHEMBL10310070 0.77 CYP2D6 (0.36) PDE2AIDO1GAATRPA1AKR1C3
SCHEMBL21457919 0.76 IDO1 (0.40) IDO1CES2PTPN5CYP3A4TSHR
SCHEMBL18242209 0.75 ERN1 (0.33) CES2
SCHEMBL28117463 0.75 PDE2A (0.49) PDE2AIDO1GAA
SCHEMBL9341736 0.74 CYP2D6 (0.39) PDE2AIDO1GAACES2CYP3A4
SCHEMBL15157741 0.72 CES2 (0.38) PDE2AIDO1GAACES2APP
SCHEMBL16327958 0.70 PDE2A (0.41) PDE2AIDO1GAACES2TSHR
SCHEMBL23571233 0.70 PDE2A (0.40) PDE2AIDO1TRPA1AKR1C3AKR1C2
SCHEMBL2005442 0.69 CES2 (0.40) PDE2AIDO1CES2PTPN5CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104169281-B The pyrroles's diformamide condensed and they are as the purposes of medicine 赛诺菲 2016-12-14 CN claimed
CN-104169281-B The pyrroles's diformamide condensed and they are as the purposes of medicine 赛诺菲 2016-12-14 CN disclosed