SCHEMBL28118959

SCHEMBL28118959

CC=NNc1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
ALDH1A1 P00352 4/20 0.46
HPGD P15428 3/20 0.46
TSHR P16473 2/20 0.46
HSD17B10 Q99714 2/20 0.46
CYP3A4 P08684 2/20 0.46
TP53 P04637 1/20 0.46
ALOX15 P16050 1/20 0.46
CDC25B P30305 1/20 0.46
ATM Q13315 1/20 0.46
KDM4E B2RXH2 4/20 0.43
GAA P10253 3/20 0.43
CA12 O43570 2/20 0.42
CA4 P22748 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
CA3 P07451 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13624676 1.00 KEAP1 (0.46) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL11433940 0.78 NOX1 (0.53) ALDH1A1HPGDTSHRHSD17B10CYP3A4
SCHEMBL3842734 0.74 KDM4E (0.52) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL9055550 0.74 ALDH1A1 (0.50) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL1342156 0.74 ALDH1A1 (0.50) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL19559633 0.74 MAPT (0.56) ALDH1A1HPGDTSHRALOX15KDM4E
SCHEMBL11433264 0.73 MAPT (0.54) ALDH1A1HPGDTSHRHSD17B10CYP3A4
SCHEMBL13875564 0.73 MAPT (0.57) ALDH1A1HPGDCYP3A4KDM4EGAA
SCHEMBL1755252 0.70 KEAP1 (0.43) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL7483801 0.70 ALDH1A1 (0.56) KEAP1ALDH1A1HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106414468-B Fumaric acid-CO- discharges molecular hybridization object, its purposes and preparation method in treatment inflammatory or cardiovascular disease 巴黎第十二大学 2019-05-03 CN disclosed
CN-106414468-A Fumarate-co-releasing molecule hybrids, their use in the treatment of inflammatory or cardiovascular diseases and their process of preparation 巴黎第十二大学 2017-02-15 CN disclosed