SCHEMBL28122002

SCHEMBL28122002

O=C(CCl)C1=NCCc2c1[nH]c1ccccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.54
MEN1 O00255 7/20 0.54
KDM4E B2RXH2 6/20 0.54
MAPT P10636 5/20 0.54
ADRB2 P07550 2/20 0.54
HTR7 P34969 2/20 0.54
POLB P06746 1/20 0.54
HTR1A P08908 1/20 0.54
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
HTR5A P47898 1/20 0.54
HTR6 P50406 1/20 0.54
NISCH Q9Y2I1 1/20 0.54
ATM Q13315 1/20 0.46
ALDH1A1 P00352 4/20 0.46
LMNA P02545 2/20 0.46
RAB9A P51151 2/20 0.46
MITF O75030 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GPX4 P36969 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27594856 0.83 MEN1 (0.59) KMT2AMEN1KDM4EMAPTADRB2
SCHEMBL6377997 0.78 KDM4E (0.57) KMT2AMEN1KDM4EMAPTADRB2
SCHEMBL6376821 0.78 AURKA (0.60) KMT2AMEN1KDM4EMAPTADRB2
Hydrochloric Acid SCHEMBL2274556 0.74 MEN1 (0.64) KMT2AMEN1KDM4EMAPTADRB2
SCHEMBL29986234 0.71 KDM4E (0.55) KMT2AMEN1KDM4EMAPTADRB2
SCHEMBL141724 0.70 MEN1 (1.00) KMT2AMEN1KDM4EMAPTADRB2
SCHEMBL9480941 0.70 MEN1 (1.00) KMT2AMEN1KDM4EMAPTADRB2
SCHEMBL6370032 0.70 MEN1 (0.55) KMT2AMEN1KDM4EMAPTADRB2
SCHEMBL2770168 0.70 MEN1 (0.65) KMT2AMEN1KDM4EMAPTADRB2
SCHEMBL27594857 0.70 MEN1 (0.55) KMT2AMEN1KDM4EMAPTADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106432234-A Method for preparing 1-phenylacetyl-beta-carboline derivatives 中国药科大学 2017-02-22 CN disclosed