SCHEMBL28124188

SCHEMBL28124188

CNc1cc2cnccc2[nH]c1=O

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.59
PDE3B Q13370 1/20 0.49
PDE3A Q14432 1/20 0.49
PARP1 P09874 4/20 0.41
HRH4 Q9H3N8 1/20 0.41
CHUK O15111 1/20 0.40
KDM5A P29375 2/20 0.40
MAPT P10636 1/20 0.40
SNCA P37840 1/20 0.40
KDM4C Q9H3R0 1/20 0.39
CNR2 P34972 1/20 0.39
NAMPT P43490 3/20 0.38
CYP2C9 P11712 2/20 0.38
CSNK2A1 P68400 1/20 0.37
AOC1 P19801 2/20 0.37
AOC3 Q16853 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7380955 0.78 DAO (0.65) DAOPDE3BPDE3APARP1HRH4
SCHEMBL12909532 0.76 BRD4 (0.59) DAOMAPTAOC3
SCHEMBL19362482 0.76 DAO (0.49) DAOPDE3BPDE3AHRH4CHUK
SCHEMBL24312093 0.75 DAO (0.61) DAOPDE3BPDE3APARP1HRH4
SCHEMBL21957317 0.75 DAO (0.65) DAOPDE3BPDE3APARP1HRH4
SCHEMBL31475468 0.75 DAO (0.65) DAOPDE3BPDE3APARP1HRH4
SCHEMBL3360519 0.75 DAO (1.00) DAOPDE3BPDE3APARP1HRH4
SCHEMBL22017082 0.74 DAO (0.59) DAOPDE3BPDE3APARP1HRH4
SCHEMBL4310842 0.74 DAO (0.59) DAOPDE3BPDE3APARP1HRH4
SCHEMBL22016192 0.74 DAO (0.59) DAOPDE3BPDE3APARP1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459034-B Carbostyril derivative as fibroblast growth factor acceptor inhibitor 普林斯匹亚生物制药公司 2018-01-12 CN disclosed
CN-106459034-A Quinolone derivatives as fibroblast growth factor receptor inhibitors 普林斯匹亚生物制药公司 2017-02-22 CN disclosed