SCHEMBL28126337

SCHEMBL28126337

C#Cc1cccc(Nc2ccc3ccccc3n2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.52
RHOA P61586 1/20 0.51
NCF1 P14598 1/20 0.45
CSNK2A2 P19784 4/20 0.44
CSNK2B P67870 4/20 0.44
CSNK2A1 P68400 4/20 0.44
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 2/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
GAA P10253 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
EGFR P00533 5/20 0.42
PDGFRB P09619 1/20 0.42
KDR P35968 1/20 0.42
KMT2A Q03164 2/20 0.42
IDO1 P14902 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29355413 0.78 ABCG2 (0.64) ABCG2CSNK2A2CSNK2BCSNK2A1ALDH1A1
SCHEMBL17432179 0.78 ABCG2 (0.64) ABCG2CSNK2A2CSNK2BCSNK2A1ALDH1A1
SCHEMBL396525 0.77 NCF1 (0.61) RHOANCF1CSNK2A1ALDH1A1KDM4E
SCHEMBL29833517 0.77 NCF1 (0.61) RHOANCF1CSNK2A1ALDH1A1KDM4E
SCHEMBL1701970 0.77 NPC1 (0.61) ABCG2RHOANCF1ALDH1A1KDM4E
SCHEMBL3951916 0.77 IGF1R (0.55) ABCG2RHOANCF1ALDH1A1KDM4E
SCHEMBL26545887 0.75 IDO1 (0.47) ABCG2CSNK2A2CSNK2BCSNK2A1ALDH1A1
SCHEMBL22627074 0.74 ABCG2 (0.51) ABCG2RHOACSNK2A2CSNK2BCSNK2A1
SCHEMBL2849200 0.74 TLR4 (0.47) ABCG2ALDH1A1EGFRPDGFRBKDR
SCHEMBL4214745 0.73 AURKA (0.58) ABCG2RHOAALDH1A1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104530061-B Icotinib hydrochloride crystal forms, medicine composition and application of icotinib hydrochloride crystal forms 贝达药业股份有限公司 2017-05-10 CN disclosed
CN-104592242-B Icotinib hydrochloride crystal forms, medicine composition and application 贝达药业股份有限公司 2017-01-25 CN disclosed