SCHEMBL28126398

SCHEMBL28126398

COc1ccc(O)c(I)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
NNMT P40261 2/20 0.39
ERN1 O75460 2/20 0.37
CYP1A2 P05177 2/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B1 P14061 2/20 0.35
HSD17B2 P37059 2/20 0.35
DYRK1A Q13627 3/20 0.35
RAF1 P04049 2/20 0.35
MAOB P27338 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA13 Q8N1Q1 1/20 0.34
MTNR1A P48039 5/20 0.33
MTNR1B P49286 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28935930 0.77 POLB (0.42) POLBTDP1NNMTERN1CYP1A2
SCHEMBL29091456 0.77 POLB (0.42) POLBTDP1NNMTERN1CYP1A2
SCHEMBL586103 0.76 NNMT (0.53) POLBTDP1NNMTERN1CYP1A2
SCHEMBL323351 0.76 POLB (0.55) POLBTDP1NNMTERN1CYP1A2
SCHEMBL30619421 0.74 POLB (0.40) POLBTDP1NNMTERN1CYP1A2
SCHEMBL3099634 0.74 NNMT (0.39) POLBTDP1NNMTCYP1A2SIRT2
SCHEMBL13213488 0.74 POLB (0.40) POLBTDP1NNMTERN1CYP1A2
SCHEMBL15467080 0.74 POLB (0.40) POLBTDP1NNMTERN1CYP1A2
SCHEMBL30427669 0.74 NNMT (0.43) POLBTDP1NNMTERN1CYP1A2
SCHEMBL20613046 0.71 KMT2A (0.45) POLBTDP1NNMTERN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108164513-A Substituted oxo pyridine derivative and its purposes in terms of cardiovascular disorder is treated 拜耳制药股份公司 2018-06-15 CN disclosed
CN-105164122-B Substituted oxopyridine derivatives and their use in the treatment of cardiovascular disorders 拜耳制药股份公司 2018-02-02 CN disclosed
CN-105849109-B Substituted oxopyridine derivatives 拜耳制药股份公司 2018-01-23 CN disclosed
CN-106687458-A Substituted oxopyridine derivatives 拜耳制药股份公司 2017-05-17 CN disclosed