SCHEMBL28127482

SCHEMBL28127482

CCOC(=O)c1cc2c3ccccc3n(Cc3ccccc3)c2c(-c2ccc(OC)c(OC)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
HTT P42858 2/20 0.46
KDM4E B2RXH2 2/20 0.46
LMNA P02545 2/20 0.46
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.45
F2RL3 Q96RI0 2/20 0.45
MAPT P10636 3/20 0.42
CNR2 P34972 1/20 0.42
TP53 P04637 1/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
PLA2G10 O15496 1/20 0.42
PLA2G1B P04054 1/20 0.42
PLA2G2A P14555 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28127494 0.91 ALDH1A1 (0.46) HTTKDM4EALDH1A1MAPTCNR2
SCHEMBL28127413 0.90 CNR2 (0.46) PDE4APDE4BPDE4CPDE4DHTT
SCHEMBL28127530 0.88 CNR2 (0.53) HTTKDM4ELMNAALDH1A1SMN1; SMN2
SCHEMBL28379309 0.87 F2RL3 (0.50) KDM4ELMNAALDH1A1F2RL3MAPT
SCHEMBL2214591 0.82 GAA (0.50) KDM4ELMNAALDH1A1F2RL3MAPT
SCHEMBL28127173 0.81 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DHTT
SCHEMBL28376283 0.80 MDM2 (0.54) HTTKDM4EALDH1A1SMN1; SMN2RXFP1
SCHEMBL28127171 0.80 KDM4E (0.52) KDM4ELMNAALDH1A1F2RL3CNR2
SCHEMBL28376586 0.79 GABRA2 (0.48) HTTKDM4EALDH1A1MAPTCNR2
SCHEMBL2216447 0.78 CNR2 (0.49) PDE4APDE4BPDE4CPDE4DKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106349257-B The double B-carboline alkaloid compounds and its pharmaceutical applications that 3 piperazine bridgings connect 新疆华世丹药物研究有限责任公司 2019-07-12 CN disclosed
CN-106349257-A 3-bit piperazine bridge connected di-beta-carboline alkali type compound and pharmaceutical application thereof 新疆华世丹药物研究有限责任公司 2017-01-25 CN disclosed