SCHEMBL28129456

SCHEMBL28129456

O=COCc1ccc(OC(F)F)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 1/20 0.41
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
DRD1 P21728 1/20 0.39
RXRA P19793 9/20 0.36
GRIN1 Q05586 9/20 0.36
GRIN2B Q13224 9/20 0.36
ALKBH1 Q13686 1/20 0.35
ATP4A P20648 1/20 0.34
ATP4B P51164 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28114840 0.79 NAAA (0.40) MBOAT4NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL21081076 0.78 DRD1 (0.49) DRD1ALKBH1MRGPRX4NPC1RAB9A
SCHEMBL28818088 0.76 DAO (0.32)
SCHEMBL29974801 0.75 MBOAT4 (0.42) MBOAT4HCRTR1HCRTR2DRD1RXRA
SCHEMBL19555693 0.75 MBOAT4 (0.45) MBOAT4HCRTR1HCRTR2DRD1RXRA
SCHEMBL4535683 0.75 MBOAT4 (0.42) MBOAT4HCRTR1HCRTR2DRD1RXRA
SCHEMBL18378650 0.75 MBOAT4 (0.45) MBOAT4HCRTR1HCRTR2RXRAGRIN1
SCHEMBL2895609 0.75 MBOAT4 (0.42) MBOAT4HCRTR1HCRTR2RXRAGRIN1
SCHEMBL28088981 0.74 BRD4 (0.35) ALDH1A1KDM4E
SCHEMBL30106088 0.73 ATM (0.44) MBOAT4HCRTR1HCRTR2ALKBH1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459088-A 2-amino-6-methyl-4,4a,5,6-tetrahydropyrano[3,4-d][1,3]thiazin-8a(8h)-yl-1,3-thiazol-4-yl amides 辉瑞公司 2017-02-22 CN disclosed