SCHEMBL28129591

SCHEMBL28129591

C=C=C.O=C(O)N1CCCc2cc(C(F)(F)F)ccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.58
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
LMNA P02545 2/20 0.44
NR3C1 P04150 1/20 0.42
NR1H3 Q13133 1/20 0.42
RAB9A P51151 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
GPBAR1 Q8TDU6 1/20 0.41
KDM4E B2RXH2 1/20 0.41
NPSR1 Q6W5P4 2/20 0.40
MAPT P10636 2/20 0.40
HSD17B10 Q99714 1/20 0.40
NPC1 O15118 1/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PDK1 Q15118 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7552151 0.95 NOTUM (0.63) NOTUMHTR2AHTR2CLMNANR3C1
SCHEMBL7382818 0.91 NOTUM (0.62) NOTUMHTR2AHTR2CLMNANR3C1
SCHEMBL30681440 0.86 NOTUM (0.76) NOTUMHTR2AHTR2CLMNACYP2C9
SCHEMBL27544652 0.83 CNR2 (0.53) NOTUMHTR2AHTR2CRAB9AHDAC1
SCHEMBL24011079 0.82 NOTUM (0.84) NOTUMLMNAMAPTL3MBTL1HTT
SCHEMBL3653813 0.79 NOTUM (0.61) NOTUMHTR2AHTR2CLMNAKDM4E
SCHEMBL26763830 0.79 NOTUM (0.61) NOTUMHTR2AHTR2CLMNANR3C1
SCHEMBL5696394 0.77 NOTUM (0.59) NOTUMHTR2AHTR2CLMNANR3C1
SCHEMBL6752845 0.77 NOTUM (0.59) NOTUMHTR2AHTR2CLMNANR3C1
SCHEMBL30767099 0.77 NOTUM (0.59) NOTUMHTR2AHTR2CLMNANR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106456539-A pharmaceutical compositions of hydrophobic compounds 阿森迪亚制药有限责任公司 2017-02-22 CN disclosed