SCHEMBL28130595

SCHEMBL28130595

Clc1ccccc1-c1ccc2c(c1)c(NC1CCNCC1)nn2Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 0.62
CLK4 Q9HAZ1 6/20 0.62
CYP2C19 P33261 5/20 0.62
CYP2D6 P10635 4/20 0.62
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
HSD17B10 Q99714 3/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 2/20 0.45
TP53 P04637 1/20 0.45
CYP2C9 P11712 1/20 0.45
MAPK14 Q16539 3/20 0.43
MAPK13 O15264 2/20 0.43
MAPK12 P53778 2/20 0.43
MAPK11 Q15759 2/20 0.43
TSHR P16473 1/20 0.43
CYP3A4 P08684 3/20 0.42
PAK4 O96013 1/20 0.39
PAK1 Q13153 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16636882 0.68 CYP1A2 (0.53) CYP1A2CLK4CYP2C19CYP2D6MEN1
SCHEMBL30608214 0.64 CYP1A2 (0.50) CYP1A2CLK4CYP2C19CYP2D6MEN1
SCHEMBL30608213 0.64 CYP1A2 (0.50) CYP1A2CLK4CYP2C19CYP2D6MEN1
SCHEMBL29102565 0.64 CYP1A2 (0.50) CYP1A2CLK4CYP2C19CYP2D6MEN1
SCHEMBL83169 0.62 CYP1A2 (0.48) CYP1A2CLK4CYP2C19CYP2D6MEN1
SCHEMBL4735299 0.62 SFRP1 (0.54) CYP1A2CLK4CYP2C19CYP2D6MEN1
SCHEMBL12277211 0.62 CYP1A2 (0.55) CYP1A2CLK4CYP2C19CYP2D6MEN1
Hydrochloric Acid SCHEMBL2418315 0.61 CYP1A2 (0.54) CYP1A2CLK4CYP2C19CYP2D6MEN1
Hydrochloric Acid SCHEMBL68901 0.61 CYP1A2 (0.47) CYP1A2CLK4CYP2C19CYP2D6MEN1
SCHEMBL26391736 0.61 CYP1A2 (0.39) CYP1A2CLK4CYP2C19CYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106488910-A Inhibitors of kras g12c 亚瑞克西斯制药公司 2017-03-08 CN disclosed