Ifetroban

Ifetroban

SCHEMBL28135

CCCCCNC(=O)c1coc([C@H]2[C@@H](Cc3ccccc3CCC(=O)O)[C@@H]3CC[C@H]2O3)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 19/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bms-180291 SCHEMBL28137 1.00 TBXA2R (1.00) TBXA2R
Ifetroban SCHEMBL30218601 1.00 TBXA2R (1.00) TBXA2R
Bms-180291 SCHEMBL9589119 1.00 TBXA2R (1.00) TBXA2R
Bms-180291 SCHEMBL29502980 1.00 TBXA2R (1.00) TBXA2R
Bms-180291 SCHEMBL28136 1.00 TBXA2R (1.00) TBXA2R
SCHEMBL8918962 0.99 TBXA2R (1.00) TBXA2R
Ifetroban SCHEMBL16212975 0.99 TBXA2R (0.98) TBXA2R
Bms-180291 SCHEMBL16212977 0.99 TBXA2R (0.98) TBXA2R
SCHEMBL8918573 0.99 TBXA2R (1.00) TBXA2R
Bms-180291 SCHEMBL362595 0.99 TBXA2R (0.98) TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5123 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260041336-A1 PLATELET REACTIVITY EXPRESSION SCORE PREDICTS CARDIOVASCULAR RISK NEW YORK UNIVERSITY (US) 2026-02-12 US claimed
US-12527839-B2 Treatments for systemic sclerosis ACCELERON PHARMA INC. (US) 2026-01-20 US claimed
EP-4482481-B1 COMPOUNDS FOR USE IN THE TREATMENT OF DYSTROPHINOPATHIES SOM INNOVATION BIOTECH S A (ES) 2025-11-12 EP claimed
US-20250152567-A1 COMPOUNDS FOR USE IN THE TREATMENT OF DYSTROPHINOPATHIES REGENTS OF THE UNIVERSITY OF MINNESOTA 2025-05-15 US claimed
US-20250144079-A1 METHODS OF INHIBITING TUMOR METASTASIS VANDERBILT UNIVERSITY 2025-05-08 US claimed
US-20250114334-A1 Ifetroban Treatment for Systemic Sclerosis VANDERBILT UNIVERSITY 2025-04-10 US claimed
CN-119522896-A Cell stabilizer and application thereof 广州市雷德生物科技有限公司 2025-02-28 CN claimed
US-20250049764-A1 Compositions and Methods of Treating Cardiac Fibrosis with Ifetroban CUMBERLAND PHARMACEUTICALS INC. 2025-02-13 US claimed
EP-4482481-A1 COMPOUNDS FOR USE IN THE TREATMENT OF DYSTROPHINOPATHIES Som Innovation Biotech, S.L. (ES) 2025-01-01 EP claimed
US-12161632-B2 Compositions and methods of treating cardiac fibrosis with ifetroban CUMBERLAND PHARMACEUTICALS INC. (US) 2024-12-10 US claimed
EP-1156803-A1 LACTAM INHIBITORS OF FXa AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2001-11-28 EP claimed
WO-2001040231-A1 HETEROCYCLIC DIHYDROPYRIMIDINES AS POTASSIUM CHANNEL INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-06-07 WO claimed
WO-2001027107-A2 HETEROCYCLIC SODIUM/PROTON EXCHANGE INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2001-04-19 WO claimed
WO-2001021602-A1 OXA- AND THIAZOLE DERIVATIVES USEFUL AS ANTIDIABETIC AND ANTIOBESITY AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-03-29 WO claimed
WO-2000047207-A1 LACTAM INHIBITORS OF FXa AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2000-08-17 WO claimed
US-5605917-A ADMINISTERING A THROMBOXANE A2 RECEPTOR ANTAGONIST BRISTOL-MYERS SQUIBB COMPANY (US) 1997-02-25 US claimed
WO-1996017606-A1 USE OF INFLAMMATORY MODULATORS IN THE TREATMENT OF CHRONIC OR RECALCITRANT SKIN DAMAGE BRISTOL-MYERS SQUIBB COMPANY (US) 1996-06-13 WO claimed
US-5506248-A SALT OF IFETROBAN AND ONE OR MORE BASIFYING AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1996-04-09 US claimed
CN-1118254-A Pharmaceutical compositions having good dissolution properties BRISTOL MYERS SQIBB COMPANY (US) 1996-03-13 CN claimed
EP-0638310-A1 Pharmaceutical compositions containing ifetroban BRISTOL-MYERS SQUIBB COMPANY (US) 1995-02-15 EP claimed