SCHEMBL28135481

SCHEMBL28135481

FC(F)(F)c1cc(-c2cscn2)ccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 11/20 0.52
RORC P51449 1/20 0.44
SCN9A Q15858 1/20 0.43
CYP1A2 P05177 1/20 0.43
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
CASP3 P42574 1/20 0.41
COMT P21964 1/20 0.41
FAAH O00519 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
MPL P40238 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15943367 0.80 AHR (0.48)
SCHEMBL28184793 0.79 CYP11B2 (0.49) SCN9AMPL
SCHEMBL14754382 0.79 KMO (0.47) RORCSCN9A
SCHEMBL28185438 0.76 SCN9A (0.44) RORCSCN9ACTSSCTSKMPL
SCHEMBL4524262 0.76 KMO (0.47) SCN9A
SCHEMBL2698021 0.75 NOTUM (0.61) NOTUMCYP1A2CASP3COMTPDE3B
SCHEMBL29699355 0.75 SCN9A (0.59) SCN9A
SCHEMBL11625443 0.74 NOTUM (0.55) NOTUMCYP1A2CTSSCTSKCASP3
SCHEMBL474200 0.74 MPL (0.71) NOTUMCASP3MPL
SCHEMBL17626005 0.74 NOTUM (0.51) NOTUMCYP1A2CTSSCTSKCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008353-B 2-acylaminothiazole derivative or salt thereof 安斯泰来制药株式会社 2017-11-10 CN disclosed
CN-106573928-A 2-aminothiazole derivative or salt thereof 安斯泰来制药株式会社 2017-04-19 CN disclosed