SCHEMBL28136347

SCHEMBL28136347

C[C](C)Cn1ccc2ccc(C(N)=O)cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
ALDH1A1 P00352 4/20 0.49
HPGD P15428 3/20 0.49
HSD17B10 Q99714 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
POLB P06746 1/20 0.49
APOBEC3A P31941 1/20 0.49
APOBEC3G Q9HC16 1/20 0.49
LMNA P02545 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27979414 0.79 MAPK1 (0.67) KDM4EALDH1A1HSD17B10SMN1; SMN2LMNA
SCHEMBL16899608 0.78 KDM4E (0.42) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL3785550 0.77 MCL1 (0.51) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL4102767 0.76 AR (0.53) KDM4EALDH1A1HSD17B10SMN1; SMN2HDAC3
SCHEMBL3429972 0.75 PLAU (0.44) KDM4EALDH1A1SMN1; SMN2POLBLMNA
SCHEMBL14632410 0.75 KMT2A (0.54) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL28116940 0.74 LCK (0.47) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
Hydrochloric Acid SCHEMBL14632367 0.74 KMT2A (0.53) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL27602860 0.73 KMT2A (0.65) LMNAKMT2A
SCHEMBL233310 0.73 HDAC11 (0.50) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104507942-B Pyridopyrimidine derivatives as protein kinase inhibitors 默克专利股份公司 2017-03-22 CN disclosed