SCHEMBL28137141

SCHEMBL28137141

COc1cc(C2=CC=NCC2)ccc1NC(=O)OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.45
SRC P12931 1/20 0.45
KDR P35968 1/20 0.45
LIMK1 P53667 1/20 0.45
LIMK2 P53671 1/20 0.45
TEK Q02763 1/20 0.45
KMT2A Q03164 4/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
HRH3 Q9Y5N1 1/20 0.44
TACR3 P29371 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
ACHE P22303 2/20 0.43
MGLL Q99685 3/20 0.41
ALDH1A1 P00352 1/20 0.41
FAAH O00519 1/20 0.41
MEN1 O00255 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HDAC3 O15379 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28328509 0.81 LCK (0.44) LCKSRCKDRLIMK1LIMK2
SCHEMBL17197477 0.78 QDPR (0.52) LCKSRCKDRLIMK1LIMK2
SCHEMBL5783658 0.74 HTT (0.59) KMT2ANPC1RAB9ATACR3CA1
SCHEMBL9524227 0.74 NPC1 (0.56) LCKSRCKDRLIMK1LIMK2
SCHEMBL17197481 0.73 HRH3 (0.49) LCKSRCKDRLIMK1LIMK2
SCHEMBL17197366 0.73 NAMPT (0.51) LCKSRCKDRLIMK1LIMK2
SCHEMBL29950865 0.72 NPC1 (0.53) KMT2ANPC1RAB9ATACR3CA1
SCHEMBL10163089 0.71 KMT2A (0.58) KMT2ANPC1RAB9ATACR3CA1
SCHEMBL9524084 0.70 LMNA (0.71) KMT2AALDH1A1MEN1HTT
SCHEMBL10929623 0.70 KMT2A (0.54) KMT2ANPC1RAB9ATACR3CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106536503-A Tyrosine kinase inhibitor and uses thereof 山东轩竹医药科技有限公司 2017-03-22 CN disclosed