SCHEMBL28137252

SCHEMBL28137252

Cc1noc(C(=O)Nc2scnc2C(N)=O)n1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 2/20 0.37
BACE1 P56817 3/20 0.36
TBK1 Q9UHD2 3/20 0.36
IKBKE Q14164 2/20 0.36
IRAK4 Q9NWZ3 1/20 0.35
FABP4 P15090 1/20 0.35
FABP5 Q01469 1/20 0.35
MAPT P10636 2/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
LMNA P02545 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18336393 0.80 TNIK (0.38) TNIKBACE1TBK1IKBKEFABP4
SCHEMBL20424077 0.73 KDM4E (0.37)
SCHEMBL20436823 0.71 KMT2A (0.51) ALDH1A1HSD17B10
SCHEMBL18337002 0.69 FABP4 (0.32) BACE1IRAK4FABP4FABP5MAPT
SCHEMBL4832820 0.69
SCHEMBL28323154 0.68 PIK3CG (0.37) BACE1IRAK4FABP4FABP5MAPT
SCHEMBL19385549 0.68 NNMT (0.38) ALDH1A1LMNAACHE
SCHEMBL8002161 0.68 KDM4E (0.49) BACE1IRAK4MAPTALDH1A1
SCHEMBL18336097 0.68 FABP4 (0.33) IRAK4FABP4FABP5ALOX15
SCHEMBL18336602 0.67 HSP90AB1 (0.33) BACE1FABP4FABP5MAPTUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106661017-A novel bicyclic or tricyclic heterocyclic compounds 田边三菱制药株式会社 2017-05-10 CN disclosed