SCHEMBL2813755

SCHEMBL2813755

CC(=O)O[C@H]1C=C[C@@](C)(O)C1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 1/20 0.33
ESR1 P03372 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MET P08581 4/20 0.33
CA12 O43570 4/20 0.33
CA9 Q16790 4/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CYP17A1 P05093 1/20 0.31
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2813758 1.00 TSHR (0.35) TSHRKMT2AALDH1A1ESR1HSD17B10
SCHEMBL30897118 0.77 CA12 (0.33) TSHRKMT2ACA12CA9CA1
SCHEMBL18306706 0.73 NPC1 (0.31) TSHRKMT2ACA12CA9CA1
SCHEMBL2816219 0.72 POLA1 (0.33) ALDH1A1CA12CA9
SCHEMBL2816300 0.72 CA12 (0.31) CA12CA9CA1CA2
SCHEMBL2816221 0.72 POLA1 (0.33) ALDH1A1CA12CA9
SCHEMBL8354298 0.68 CA12 (0.42) TSHRKMT2AALDH1A1CA12CA9
SCHEMBL11548381 0.68 CA12 (0.42) TSHRKMT2ACA12CA9CA1
SCHEMBL11548379 0.68 CA12 (0.42) TSHRKMT2ACA12CA9CA1
SCHEMBL2290500 0.68 CA12 (0.42) TSHRKMT2ACA12CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8318804-B2 Antiviral activity of cyclopentene nitro-ester and derivatives UNIVERSITY OF SOUTH FLORIDA (US) 2012-11-27 US disclosed
US-8236853-B1 Formation of cyclopentene nitro-ester and derivatives UNIVERSITY OF SOUTH FLORIDA (US) 2012-08-07 US disclosed
US-8236853-B1 Formation of cyclopentene nitro-ester and derivatives UNIVERSITY OF SOUTH FLORIDA (US) 2012-08-07 US disclosed
US-20100249230-A1 ANTIVIRAL ACTIVITY OF CYCLOPENTENE NITRO-ESTER AND DERIVATIVES UNIVERSITY OF SOUTH FLORIDA (US) 2010-09-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100249230-A1 ANTIVIRAL ACTIVITY OF CYCLOPENTENE NITRO-ESTER AND DERIVATIVES CYP51A1, CES2, DDT TSHR 4423/4885KMT2A 4206/4885ALDH1A1 1609/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.