SCHEMBL28137652

SCHEMBL28137652

Cn1c(=O)c2[nH]cnc2n(C(F)F)c1=O

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 9/20 0.75
ATAD2 Q6PL18 1/20 0.66
PDE4A P27815 10/20 0.64
PDE4B Q07343 10/20 0.64
PDE4C Q08493 10/20 0.64
PDE4D Q08499 10/20 0.64
ADORA2A P29274 9/20 0.64
ADORA3 P0DMS8 4/20 0.64
ADORA1 P30542 2/20 0.64
PIK3CD O00329 1/20 0.64
ALPL P05186 1/20 0.64
TMIGD3 P0DMS9 1/20 0.64
CYP2C19 P33261 1/20 0.64
HIF1A Q16665 1/20 0.64
CYP1A2 P05177 2/20 0.61
CFTR P13569 2/20 0.61
MAPK1 P28482 2/20 0.61
PDE2A O00408 1/20 0.61
PDE5A O76074 1/20 0.61
CYP3A4 P08684 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23073728 0.86 ADORA2B (1.00) ADORA2BATAD2PDE4APDE4BPDE4C
SCHEMBL295963 0.83 ADORA2B (0.78) ADORA2BATAD2PDE4APDE4BPDE4C
SCHEMBL7554983 0.81 ADORA2B (0.74) ADORA2BATAD2PDE4APDE4BPDE4C
Theophylline Anhydrous SCHEMBL28323421 0.80 ATAD2 (0.93) ADORA2BATAD2PDE4APDE4BPDE4C
Theophylline Anhydrous SCHEMBL28870701 0.80 ADORA2B (0.83) ADORA2BATAD2PDE4APDE4BPDE4C
Theophylline Anhydrous SCHEMBL4915 0.80 ATAD2 (1.00) ADORA2BATAD2PDE4APDE4BPDE4C
Theophylline Anhydrous SCHEMBL8595167 0.80 ATAD2 (1.00) ADORA2BATAD2PDE4APDE4BPDE4C
Theophylline Anhydrous SCHEMBL25398274 0.80 ATAD2 (1.00) ADORA2BATAD2PDE4APDE4BPDE4C
Theophylline Anhydrous SCHEMBL3051675 0.80 ATAD2 (1.00) ADORA2BATAD2PDE4APDE4BPDE4C
SCHEMBL27620327 0.79 ATAD2 (0.72) ADORA2BATAD2PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106573934-B The inhibition of transient receptor potential A1 ion channel 伊莱利利公司 2019-10-11 CN disclosed
CN-106573934-A Inhibiting the transient receptor potential A1 ion channel 海德拉生物科学公司 2017-04-19 CN disclosed