SCHEMBL28138388

SCHEMBL28138388

c1ccc(C2CN(c3ccccc3)C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BPTF Q12830 1/20 0.52
BRD4 O60885 3/20 0.42
SLC18A3 Q16572 2/20 0.42
SIGMAR1 Q99720 2/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
ADRB1 P08588 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
LMNA P02545 1/20 0.41
NOTUM Q6P988 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
SRD5A1 P18405 1/20 0.40
MBTD1 Q05BQ5 1/20 0.39
L3MBTL3 Q96JM7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31224856 0.86 MAPT (0.42) BPTFBRD4SLC18A3LMNAGAA
SCHEMBL16669158 0.83 NOTUM (0.53) SLC18A3NOTUMMAPTMBTD1L3MBTL3
SCHEMBL2725262 0.80 FFAR4 (0.56) SLC18A3NOTUMDRD2DRD4
SCHEMBL31224958 0.78 MAPT (0.51) ADRB1LMNAGAAMAPTL3MBTL1
SCHEMBL7446491 0.77 MBTD1 (0.55) SLC18A3SIGMAR1HTR3EHTR3BADRB1
SCHEMBL5537574 0.76 BPTF (0.47) BPTFSLC18A3SIGMAR1HTR3EHTR3B
SCHEMBL11696584 0.76 G6PD (0.47) BPTFBRD4SLC18A3SIGMAR1GAA
SCHEMBL23978897 0.73 BRD4 (0.44) BRD4SLC18A3SIGMAR1DRD2DRD4
SCHEMBL3121777 0.73 BPTF (0.54) BPTFSIGMAR1HTR3EHTR3BADRB1
SCHEMBL2330436 0.73 BPTF (0.54) BPTFSIGMAR1HTR3EHTR3BADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104703987-B PDE9 inhibitors having an imidazopyrazinone backbone H.隆德贝克有限公司 2017-05-03 CN claimed