SCHEMBL28141663

SCHEMBL28141663

CCN(C)S(=O)(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
LSS P48449 4/20 0.49
TRPV4 Q9HBA0 1/20 0.49
LMNA P02545 2/20 0.48
HTT P42858 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
KDM4E B2RXH2 1/20 0.48
GAA P10253 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MMP3 P08254 1/20 0.46
KIF11 P52732 2/20 0.44
NR1H3 Q13133 1/20 0.44
VCAM1 P19320 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16508752 0.86 HTR2A (0.48) HTR2AHTR2CLSSTRPV4LMNA
SCHEMBL28035458 0.84 HTT (0.63) HTR2AHTR2CLMNAHTTSMN1; SMN2
SCHEMBL16508863 0.83 LSS (0.48) HTR2AHTR2CLSSTRPV4LMNA
SCHEMBL13465623 0.81 TRPV4 (0.67) HTR2AHTR2CTRPV4LMNAHTT
SCHEMBL10263936 0.79 KMT2A (0.57) LMNAHTTSMN1; SMN2KDM4EGAA
SCHEMBL12571055 0.79 HDAC4 (0.48) HTR2AHTR2CLSSTRPV4LMNA
SCHEMBL6018716 0.79 LSS (0.58) HTR2AHTR2CLSSTRPV4
SCHEMBL6018713 0.79 LSS (0.58) HTR2AHTR2CLSSTRPV4
SCHEMBL28035878 0.78 HTR2A (0.53) HTR2AHTR2CLSSTRPV4MMP3
SCHEMBL13434084 0.77 MAPT (0.57) LMNAHTTSMN1; SMN2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106986857-B Trk inhibiting compound 小野药品工业株式会社 2019-07-05 CN disclosed
CN-106986857-A Trk inhibiting compounds 小野药品工业株式会社 2017-07-28 CN disclosed
CN-106928197-A Trk inhibiting compounds 小野药品工业株式会社 2017-07-07 CN disclosed
CN-104995172-B Trk inhibiting compounds 小野药品工业株式会社 2017-05-31 CN disclosed