SCHEMBL28035458

SCHEMBL28035458

CCN(CC)S(=O)(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 7/20 0.63
LMNA P02545 6/20 0.63
SMN1; SMN2 Q16637 5/20 0.63
NPSR1 Q6W5P4 3/20 0.59
GAA P10253 2/20 0.59
KDM4E B2RXH2 1/20 0.59
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58
MAPT P10636 2/20 0.56
PTGDR2 Q9Y5Y4 1/20 0.54
MMP3 P08254 1/20 0.54
ABCC9 O60706 1/20 0.51
ABCC8 Q09428 1/20 0.51
KCNJ11 Q14654 1/20 0.51
KCNJ8 Q15842 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
XBP1 P17861 1/20 0.50
PAX8 Q06710 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27312349 0.88 HTT (0.56) HTTLMNASMN1; SMN2NPSR1GAA
SCHEMBL28141663 0.84 HTR2A (0.50) HTTLMNASMN1; SMN2NPSR1GAA
SCHEMBL14349177 0.83 HTT (0.66) HTTLMNASMN1; SMN2NPC1RAB9A
SCHEMBL4927115 0.83 HTT (0.56) HTTLMNASMN1; SMN2NPSR1GAA
SCHEMBL13465623 0.79 TRPV4 (0.67) HTTLMNASMN1; SMN2KDM4EMAPT
SCHEMBL3246445 0.79 ALDH1A1 (0.73) HTTLMNASMN1; SMN2NPC1RAB9A
SCHEMBL28340795 0.78 KEAP1 (0.49) HTTLMNASMN1; SMN2NPSR1GAA
SCHEMBL27312342 0.78 HTT (0.50) HTTLMNASMN1; SMN2NPSR1GAA
SCHEMBL16508752 0.77 HTR2A (0.48) HTTLMNASMN1; SMN2NPSR1GAA
SCHEMBL23057256 0.76 LMNA (0.73) HTTLMNASMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106986857-B Trk inhibiting compound 小野药品工业株式会社 2019-07-05 CN disclosed
CN-106986857-A Trk inhibiting compounds 小野药品工业株式会社 2017-07-28 CN disclosed
CN-106928197-A Trk inhibiting compounds 小野药品工业株式会社 2017-07-07 CN disclosed
CN-104995172-B Trk inhibiting compounds 小野药品工业株式会社 2017-05-31 CN disclosed
CN-104995172-A Trk inhibiting compounds ONO PHARMACEUTICAL CO 2015-10-21 CN disclosed