SCHEMBL2814434

SCHEMBL2814434

COCCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc([N+](=O)[O-])cc3)NC(=O)OC(C)(C)C)C2)c(C)c2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 2/20 0.39
KLK5 Q9Y337 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CNR2 P34972 2/20 0.35
ALDH1A1 P00352 1/20 0.34
ACE P12821 1/20 0.34
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
PADI4 Q9UM07 1/20 0.33
HTR2A P28223 2/20 0.33
HTR4 Q13639 2/20 0.33
SCN9A Q15858 1/20 0.32
CHRM3 P20309 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2814433 1.00 PROKR1 (0.39) PROKR1KLK5SMN1; SMN2CNR2ALDH1A1
SCHEMBL7899697 0.91 PROKR1 (0.39) PROKR1KLK5CNR2ALDH1A1ACE
SCHEMBL7891211 0.91 PROKR1 (0.42) PROKR1KLK5CNR2ALDH1A1ACE
SCHEMBL7902566 0.90 PROKR1 (0.38) PROKR1KLK5CNR2ACEHRH2
SCHEMBL7897770 0.88 PROKR1 (0.37) PROKR1KLK5CNR2ACEHRH2
SCHEMBL2788344 0.88 PROKR1 (0.38) PROKR1KLK5CNR2ALDH1A1ACE
SCHEMBL7903380 0.87 PROKR1 (0.39) PROKR1KLK5CNR2ACEHRH2
SCHEMBL2814775 0.87 PROKR1 (0.37) PROKR1KLK5CNR2ACEHRH2
SCHEMBL7893430 0.87 USP30 (0.36) PROKR1KLK5CNR2ACEHRH2
SCHEMBL2814776 0.87 PROKR1 (0.37) PROKR1KLK5CNR2ACEHRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed