SCHEMBL28144725

SCHEMBL28144725

COC(=O)c1ccc(C(F)(F)F)c(Cl)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.67
PDK2 Q15119 3/20 0.55
PDK1 Q15118 2/20 0.55
PDK3 Q15120 2/20 0.55
PDK4 Q16654 2/20 0.55
ALDH1A1 P00352 4/20 0.50
MRGPRX4 Q96LA9 2/20 0.48
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
XDH P47989 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
KDM4E B2RXH2 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47
CNR2 P34972 1/20 0.46
P4HB P07237 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL197395 0.87 NOTUM (0.62) NOTUMPDK2PDK1PDK3PDK4
SCHEMBL15077181 0.85 PDK1 (0.52) NOTUMPDK2PDK1PDK3PDK4
SCHEMBL1997248 0.84 NOTUM (0.73) NOTUMPDK2PDK1PDK3PDK4
SCHEMBL665618 0.83 CA12 (0.51) NOTUMPDK2PDK1PDK3PDK4
SCHEMBL9859293 0.81 MEN1 (0.47) NOTUMPDK2PDK1PDK3PDK4
SCHEMBL3902096 0.81 NOTUM (0.69) NOTUMPDK2ALDH1A1MRGPRX4CA12
SCHEMBL3830811 0.81 NOTUM (0.69) NOTUMPDK2ALDH1A1MRGPRX4CA12
SCHEMBL3903076 0.81 NOTUM (0.69) NOTUMPDK2PDK1PDK3PDK4
SCHEMBL536555 0.81 NOTUM (0.52) NOTUMPDK2PDK1PDK3PDK4
SCHEMBL313146 0.81 KIF11 (0.54) NOTUMPDK1MRGPRX4RAB9ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119325476-A Nitrogen-containing condensed 2, 3-dihydroquinazolinone compounds as NAV1.8 inhibitors 葛兰素史密斯克莱知识产权发展有限公司 2025-01-17 CN disclosed
CN-106794161-A TrkA kinase inhibitors, composition and its method 默沙东公司 2017-05-31 CN disclosed