SCHEMBL28145488

SCHEMBL28145488

CC(C)CN(c1ccccc1N)C1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 10/20 0.38
CCKBR P32239 1/20 0.36
KDM4E B2RXH2 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
AOC3 Q16853 1/20 0.34
LMNA P02545 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.33
USP2 O75604 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PABPC1 P11940 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13130610 0.90 KDM4E (0.34) IDO1KDM4EGAAMAPTLMNA
SCHEMBL16538494 0.80 IDO1 (0.41) IDO1SLC6A2SLC6A4LMNAMEN1
SCHEMBL20301578 0.80 IDO1 (0.35) IDO1CCKBR
SCHEMBL28094663 0.78 BCHE (0.36) KDM4EGAAMAPTLMNA
SCHEMBL20321883 0.76 IDO1 (0.39) IDO1KDM4EGAAMAPTMEN1
SCHEMBL10984066 0.76 KDM4E (0.36) KDM4EGAAMAPTLMNAMEN1
SCHEMBL28842010 0.75 THRA (0.38) KDM4EGAAMAPTHSD17B10
SCHEMBL28388284 0.75 THRA (0.38) KDM4EGAAMAPTLMNAHSD17B10
SCHEMBL4471183 0.75 CCKBR (0.39) IDO1CCKBRSLC6A2SLC6A4MEN1
SCHEMBL6254408 0.75 AOC3 (0.43) GAASLC6A2SLC6A4AOC3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658643-B IDO inhibitor 百时美施贵宝公司 2019-03-01 CN disclosed
CN-105324362-B Ido inhibitors 百时美施贵宝公司 2017-05-24 CN disclosed