SCHEMBL28147205

SCHEMBL28147205

FC(F)(F)c1ccc(-c2nc(-c3ccc(Br)cc3)n[nH]2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 5/20 0.67
NR1H3 Q13133 5/20 0.67
DGAT1 O75907 1/20 0.67
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
KDM4E B2RXH2 1/20 0.54
POLB P06746 1/20 0.54
ATM Q13315 1/20 0.54
TRPV1 Q8NER1 1/20 0.52
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
HTT P42858 1/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
AHR P35869 1/20 0.47
LMNA P02545 1/20 0.46
PLCG1 P19174 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29035846 0.86 NR1H2 (0.71) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL14521015 0.86 NR1H2 (0.71) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL26464405 0.84 NPC1 (0.67) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL11319935 0.82 NR1H2 (0.73) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL17280061 0.81 NPC1 (0.55) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL1260404 0.81 KIF11 (0.58) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL1230235 0.81 NPC1 (0.50) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL28147211 0.80 NR1H2 (1.00) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL27935074 0.80 NPC1 (0.49) NR1H2NR1H3DGAT1NPC1RAB9A
SCHEMBL15299217 0.77 AOC3 (0.52) NR1H2NR1H3DGAT1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106632106-A Synthetic method of asymmetric 1,2,4-triazole derivatives 安徽师范大学 2017-05-10 CN disclosed