SCHEMBL28149986

SCHEMBL28149986

CC(C)n1ccc(OCC(F)(F)F)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
LRRK2 Q5S007 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
DYRK1A Q13627 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 3/20 0.34
CYP17A1 P05093 2/20 0.34
CYP2C9 P11712 2/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
JMJD6 Q6NYC1 1/20 0.32
CACNA1G O43497 1/20 0.31
CACNA1H O95180 1/20 0.31
CACNA1I Q9P0X4 1/20 0.31
SCN9A Q15858 1/20 0.31
ACACB O00763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22943261 0.86 HDAC1 (0.36) HDAC1HDAC6DYRK1A
SCHEMBL17658980 0.85 NUDT1 (0.40) HDAC1HDAC6DYRK1A
SCHEMBL21468722 0.77 DYRK1A (0.37) HDAC1HDAC6DYRK1A
SCHEMBL20759271 0.77 DYRK1A (0.37) HDAC1HDAC6SMN1; SMN2L3MBTL1DYRK1A
SCHEMBL20260592 0.76 CFTR (0.35) HDAC1HDAC6ACACB
SCHEMBL21452646 0.76 DYRK1A (0.36) HDAC1HDAC6SMN1; SMN2DYRK1AACACB
SCHEMBL22943015 0.75 DYRK1A (0.36) HDAC1HDAC6DYRK1A
SCHEMBL21452644 0.74 CFTR (0.37) HDAC1HDAC6
SCHEMBL20522883 0.74 SCN9A (0.34) SMN1; SMN2L3MBTL1PTGS1PTGS2SCN9A
SCHEMBL22943016 0.73 DYRK1A (0.33) HDAC1HDAC6DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106255688-B Morpholine-pyridine derivate 豪夫迈·罗氏有限公司 2019-11-08 CN disclosed
CN-106661043-A 2-oxa-5-azabicyclo[2.2.1]heptan-3-yl derivatives 豪夫迈·罗氏有限公司 2017-05-10 CN disclosed