SCHEMBL28153158

SCHEMBL28153158

CCCN1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)OCC

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 1/20 0.39
KCNH2 Q12809 1/20 0.37
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
SLC6A2 P23975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28153157 1.00 CYP3A4 (0.44) CYP3A4MAPTALDH1A1KCNH2SLC6A4
SCHEMBL28152039 0.81 ALDH1A1 (0.43) CYP3A4MAPTALDH1A1SLC6A4SLC6A3
SCHEMBL10217221 0.78 MAPT (0.36) CYP3A4MAPTALDH1A1KCNH2
SCHEMBL4736905 0.78 MAPT (0.36) CYP3A4MAPTALDH1A1KCNH2
SCHEMBL21159397 0.77 OPRK1 (0.48) ALDH1A1KCNH2SLC6A4
SCHEMBL29638013 0.77 OPRK1 (0.48) ALDH1A1KCNH2SLC6A4
SCHEMBL15934617 0.77 OPRK1 (0.48) ALDH1A1KCNH2SLC6A4
SCHEMBL29641090 0.77 OPRK1 (0.48) ALDH1A1KCNH2SLC6A4
SCHEMBL29641135 0.77 OPRK1 (0.48) ALDH1A1KCNH2SLC6A4
SCHEMBL9082047 0.77 ALDH1A1 (0.37) MAPTALDH1A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106928127-B Substituted piperidine amide derivative, preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2021-07-16 CN disclosed
CN-106928127-A Substituted piperidine class amide derivatives and preparation method thereof and application pharmaceutically 四川海思科制药有限公司 2017-07-07 CN disclosed