SCHEMBL28158441

SCHEMBL28158441

NC(=O)c1cc(C2CC2)nn1Cl

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.34
CYP3A4 P08684 1/20 0.34
GAA P10253 1/20 0.34
CYP2C19 P33261 1/20 0.34
RET P07949 1/20 0.34
PARP1 P09874 4/20 0.33
PARP2 Q9UGN5 4/20 0.33
PSMB8 P28062 1/20 0.33
PSMB9 P28065 1/20 0.33
PSMB5 P28074 1/20 0.33
KCNJ6 P48051 3/20 0.32
KCNJ5 P48544 3/20 0.32
KCNJ3 P48549 3/20 0.32
CRACR2A Q9BSW2 1/20 0.32
KCNT1 Q5JUK3 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28149980 0.86 POLB (0.37) CYP3A4GAACYP2C19KCNJ6KCNJ5
SCHEMBL4072006 0.81 PSMB8 (0.45) SRCCYP3A4GAACYP2C19RET
SCHEMBL28157869 0.81 SRC (0.34) SRCCYP3A4GAACYP2C19RET
SCHEMBL27836331 0.77 RET (0.47) RETPSMB8PSMB9PSMB5KCNT1
SCHEMBL4069114 0.74 KCNJ6 (0.53) GAAPARP1PARP2KCNJ6KCNJ5
SCHEMBL27028207 0.72 PARP1 (0.40) PARP1PARP2PSMB8PSMB9PSMB5
SCHEMBL30559538 0.72 KCNJ6 (0.39) RETPARP1PSMB8PSMB9PSMB5
SCHEMBL3065968 0.70 KCNT1 (0.46) CYP3A4GAACYP2C19PSMB8PSMB9
SCHEMBL26976565 0.69 PDK1 (0.41) CYP3A4GAACYP2C19PSMB8PSMB9
SCHEMBL15718192 0.68 SRC (0.36) SRCRETPARP1CRACR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107001259-A Substituted azetidine derivatives as TAAR ligands 豪夫迈·罗氏有限公司 2017-08-01 CN claimed
CN-107001259-A Substituted azetidine derivatives as TAAR ligands 豪夫迈·罗氏有限公司 2017-08-01 CN disclosed