SCHEMBL28158644

SCHEMBL28158644

CCCNc1cc(Cl)ncn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNM2 P50570 2/20 0.45
NPC1 O15118 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
EGFR P00533 1/20 0.40
HTT P42858 2/20 0.38
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
HCAR3 P49019 1/20 0.37
TNNI3K Q59H18 1/20 0.36
POLB P06746 1/20 0.36
MKNK1 Q9BUB5 1/20 0.35
CHRM4 P08173 1/20 0.35
CDC7 O00311 1/20 0.35
ROCK2 O75116 1/20 0.35
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9181933 0.89 DNM2 (0.54) DNM2NPC1MEN1KMT2AEGFR
SCHEMBL5665700 0.87 DNM2 (0.60) DNM2NPC1MEN1KMT2AEGFR
SCHEMBL374260 0.84 EGFR (0.53) DNM2NPC1MEN1KMT2AEGFR
SCHEMBL5026959 0.81 CYP2D6 (0.54) NPC1MEN1KMT2AEGFRALDH1A1
SCHEMBL20081779 0.80 HRH3 (0.44) DNM2NPC1MEN1KMT2AEGFR
SCHEMBL16656099 0.80 CYP1A2 (0.54) NPC1MEN1KMT2AHTTALDH1A1
SCHEMBL23877916 0.80 HRH3 (0.51) DNM2NPC1MEN1KMT2AEGFR
SCHEMBL29526065 0.79 SMN1; SMN2 (0.47) DNM2NPC1MEN1KMT2AHTT
SCHEMBL15923128 0.78 DNM2 (0.55) DNM2NPC1MEN1KMT2AHTT
SCHEMBL15923413 0.78 DNM2 (0.55) DNM2NPC1MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105636958-B DNA PK inhibitor 沃泰克斯药物股份有限公司 2018-01-05 CN disclosed
CN-106986863-A DNA PK inhibitor 沃泰克斯药物股份有限公司 2017-07-28 CN disclosed
CN-106977495-A DNA PK inhibitor 沃泰克斯药物股份有限公司 2017-07-25 CN disclosed