SCHEMBL28158705

SCHEMBL28158705

CCc1c(N)nc2ccccc2c1CC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 11/20 0.56
ALDH1A1 P00352 4/20 0.53
HPGD P15428 4/20 0.53
KDM4E B2RXH2 3/20 0.53
GAA P10253 2/20 0.53
TLR7 Q9NYK1 4/20 0.51
DCPS Q96C86 1/20 0.47
HSD17B10 Q99714 3/20 0.47
GLA P06280 1/20 0.47
CHRM2 P08172 1/20 0.47
ADRA2A P08913 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
CHRM1 P11229 1/20 0.47
NQO2 P16083 1/20 0.47
MAOA P21397 1/20 0.47
DRD1 P21728 1/20 0.47
ACHE P22303 1/20 0.47
SLC6A2 P23975 1/20 0.47
CASP1 P29466 1/20 0.47
ADRA1A P35348 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16836314 0.85 TLR8 (0.79) TLR8ALDH1A1HPGDKDM4EGAA
SCHEMBL3343183 0.81 KDM4E (0.69) TLR8ALDH1A1HPGDKDM4EGAA
Iodide SCHEMBL10800767 0.79 KDM4E (0.67) TLR8ALDH1A1HPGDKDM4EGAA
SCHEMBL14533471 0.77 KDM4E (0.53) TLR8ALDH1A1HPGDKDM4EGAA
SCHEMBL28002147 0.77 KDM4E (0.53) ALDH1A1HPGDKDM4EGAATDP1
Ammonia Solution, Strong SCHEMBL29175740 0.77 GPR3 (0.53) TLR8ALDH1A1HPGDKDM4EGAA
SCHEMBL11703072 0.75 KDM4E (0.51) TLR8ALDH1A1HPGDKDM4EGAA
SCHEMBL6263720 0.74 TLR8 (0.82) TLR8ALDH1A1HPGDKDM4EGAA
SCHEMBL16836321 0.74 TLR8 (0.74) TLR8TLR7SMN1; SMN2
SCHEMBL16836317 0.74 TLR8 (0.65) TLR8ALDH1A1HPGDKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829294-B The quinolyl conditioning agent of ROR- γ-T being connect with methylene 詹森药业有限公司 2018-11-09 CN disclosed
CN-105209453-B The quinolyl conditioning agent of the methylene connection of ROR γ T 詹森药业有限公司 2017-06-20 CN disclosed