SCHEMBL28159262

SCHEMBL28159262

CN(C)c1nc2ccccc2cc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
ALDH1A1 P00352 4/20 0.46
HPGD P15428 3/20 0.46
MAPT P10636 3/20 0.46
GLA P06280 2/20 0.46
ACHE P22303 1/20 0.46
NCF1 P14598 1/20 0.46
KDM4E B2RXH2 4/20 0.40
CYP1A2 P05177 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
PDE10A Q9Y233 2/20 0.40
TSHR P16473 2/20 0.40
GAA P10253 1/20 0.40
STAT3 P40763 1/20 0.40
LMNA P02545 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12991538 0.78 TDP1 (0.55) TDP1ALDH1A1HPGDMAPTGLA
SCHEMBL28019424 0.74 PSMB5 (0.54) TDP1ALDH1A1HPGDMAPTGLA
SCHEMBL6849143 0.74 ALDH1A1 (0.59) TDP1ALDH1A1HPGDMAPTGLA
SCHEMBL1811989 0.74 TDP1 (0.44) TDP1ALDH1A1HPGDMAPTGLA
SCHEMBL16764607 0.73 ALDH1A1 (0.67) TDP1ALDH1A1HPGDMAPTGLA
Acridine SCHEMBL8003444 0.73 ALDH1A1 (0.71) TDP1ALDH1A1HPGDMAPTGLA
SCHEMBL2596089 0.73 TDP1 (0.63) TDP1ALDH1A1HPGDMAPTGLA
SCHEMBL30511098 0.73 TDP1 (0.63) TDP1ALDH1A1HPGDMAPTGLA
SCHEMBL22263495 0.72 PPARD (0.47) TDP1ALDH1A1HPGDMAPTGLA
SCHEMBL2487289 0.72 PPARD (0.50) ALDH1A1HPGDKDM4ESMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189498-B Geminally substituted cyanoethylpyrazolopyridinones as JANUS kinase inhibitors 默沙东公司 2017-06-27 CN disclosed