SCHEMBL28164372

SCHEMBL28164372

OC[C@H]1CC[C@H](CC(F)(F)F)CC1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.35
ESR1 P03372 6/20 0.34
ESR2 Q92731 6/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17813 0.86
SCHEMBL17388557 0.78
SCHEMBL130642 0.76 ESR2 (0.46) APLNRESR1ESR2CYP3A4CYP2C9
SCHEMBL2267415 0.76 ESR2 (0.46) APLNRESR1ESR2CYP3A4CYP2C9
SCHEMBL4610 0.76
SCHEMBL27912 0.76 ESR2 (0.46) APLNRESR1ESR2CYP3A4CYP2C9
SCHEMBL1316560 0.76 ESR2 (0.46) APLNRESR1ESR2CYP3A4CYP2C9
SCHEMBL297828 0.76 ESR2 (0.46) APLNRESR1ESR2CYP3A4CYP2C9
SCHEMBL101985 0.76 THRA (0.47) APLNRESR1ESR2CYP3A4CYP2C9
SCHEMBL1445018 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074852-B The pyrrolin and pyridine inhibitors of ROR- γ 生命医药有限责任公司 2019-08-16 CN disclosed
CN-107074852-A ROR γ pyrrolin and pyridine inhibitors 生命医药公司 2017-08-18 CN disclosed