SCHEMBL28165019

SCHEMBL28165019

NC(=O)c1cccc2ccn(C(F)(F)F)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.41
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 3/20 0.40
GAA P10253 1/20 0.40
PDPK1 O15530 1/20 0.39
PLK4 O00444 1/20 0.37
CHEK1 O14757 1/20 0.37
AURKA O14965 1/20 0.37
DAPK3 O43293 1/20 0.37
MAP4K4 O95819 1/20 0.37
CSF1R P07333 1/20 0.37
RET P07949 1/20 0.37
FGFR1 P11362 1/20 0.37
PDGFRA P16234 1/20 0.37
LTK P29376 1/20 0.37
KDR P35968 1/20 0.37
MAP2K2 P36507 1/20 0.37
FLT3 P36888 1/20 0.37
CSNK1A1 P48729 1/20 0.37
PRKX P51817 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28164511 0.85 ALDH1A1 (0.42) KDM4EALDH1A1SMN1; SMN2MAPTHPGD
SCHEMBL9275405 0.75 PARP1 (0.44) PARP1KDM4EALDH1A1GAAPDPK1
SCHEMBL30082247 0.75 PARP1 (0.44) PARP1KDM4EALDH1A1GAAPDPK1
SCHEMBL23890397 0.72 PARP1 (0.39) PARP1KDM4EALDH1A1GAAPDPK1
SCHEMBL23890365 0.71 KDM4E (0.64) PARP1KDM4EALDH1A1AURKAPARP2
SCHEMBL28193895 0.71 PARP1 (0.41) PARP1KDM4EALDH1A1GAAPDPK1
SCHEMBL22414206 0.67 FABP4 (0.43) KDM4EALDH1A1SMN1; SMN2MAPTHPGD
SCHEMBL1290332 0.66 PARP1 (0.47) PARP1KDM4EAURKA
SCHEMBL22414132 0.65 KDM4E (0.43) PARP1KDM4EALDH1A1PARP2PARP3
SCHEMBL27722750 0.65 PARP1 (0.49) PARP1KDM4EALDH1A1GAAPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110511209-A It can be used as the indole carboxamides compound of kinase inhibitor BRISTOL MYERS SQUIBB CO 2019-11-29 CN disclosed
CN-107108583-A Indole carboxamide compounds useful as kinase inhibitors 百时美施贵宝公司 2017-08-29 CN disclosed