SCHEMBL28166707

SCHEMBL28166707

NN(C(=O)O)c1ccc2[nH]ccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.46
SLC6A4 P31645 4/20 0.46
SLC6A3 Q01959 3/20 0.46
USP2 O75604 1/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 1/20 0.46
RAD51 Q06609 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CTNNB1 P35222 1/20 0.44
WNT3A P56704 1/20 0.44
F2 P00734 1/20 0.44
NPC1 O15118 2/20 0.43
MAPT P10636 2/20 0.43
RAB9A P51151 2/20 0.43
PTGS2 P35354 1/20 0.42
CYP2A6 P11509 2/20 0.42
IMPDH2 P12268 1/20 0.42
IMPDH1 P20839 1/20 0.42
AHR P35869 3/20 0.42
NR4A2 P43354 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3632143 0.83 USP2 (0.48) SLC6A2SLC6A4SLC6A3USP2GAA
SCHEMBL9717426 0.80 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3USP2GAA
SCHEMBL22418878 0.78 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3USP2GAA
SCHEMBL15253052 0.76 MAOA (0.51) SLC6A2SLC6A4SLC6A3USP2GAA
SCHEMBL8531102 0.76 NPC1 (0.43) SLC6A2SLC6A4SLC6A3USP2GAA
SCHEMBL1122014 0.75 F2 (0.46) SLC6A2SLC6A4SLC6A3USP2GAA
SCHEMBL6166853 0.75 SLC6A2 (0.48) SLC6A2SLC6A4SLC6A3USP2GAA
SCHEMBL9967028 0.74 USP2 (0.55) SLC6A2SLC6A4SLC6A3USP2GAA
SCHEMBL4362240 0.74 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3CTNNB1WNT3A
SCHEMBL28284712 0.73 CDK8 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107106700-A Peptide simulated compound and its antibody drug conjugate 基因泰克公司 2017-08-29 CN disclosed
CN-105636612-A 1- (chloromethyl) -2, 3-dihydro-1H-benzo [ e ] indole dimer antibody-drug conjugate compounds, and methods of use and treatment GENENTECH INC 2016-06-01 CN disclosed